Desfesoterodine - HY-76569

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Catalog #
HY-76569
Ab 186,00 €
Desfesoterodine (PNU-200577) is a potent and selective muscarinic receptor (mAChR) antagonist with a KB and a pA2 of 0.84 nM and 9.14, respectively[1]. Desfesoterodine is a major pharmacologically active metabolite of Tolterodine (PNU-200583; HY-A0024) and Fesoterodine (HY-70053)[2][3]. Desfesoterodine improves cerebral infarction induced detrusor overactivity in rats[4].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-76569/Desfesoterodine-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Neuroscience-Neuromodulation
Alternative Names PNU-200577; 5-Hydroxymethyl Tolterodine
CAS 207679-81-0
Storage -20°C, 3 years; 4°C, 2 years (Powder)
MWT 341.495
Solubility DMSO : 50 mg/mL (ultrasonic)|H2O : 100 mg/mL (ultrasonic)
Clinical Information Launched
Target mAChR
Applications
Application: Neuroscience-Neuromodulation

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