Lonidamine - HY-B0486

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Catalog #
HY-B0486
Ab 68,00 €
Lonidamine (AF-1890) is a hexokinase and mitochondrial pyruvate carrier inhibitor (Ki: 2.5 μM). Lonidamine also inhibits aerobic glycolysis in cancer cells. Lonidamine can be used in the research of mitochondrial metabolism and inflammation, such as pulmonary fibrosis[1][2][3].
Weitere Informationen
Datasheet URL http://file.medchemexpress.com/batch_PDF/HY-B0486/Lonidamine-DataSheet-MedChemExpress.pdf
Shipping Room Temperature
Application Cancer-Kinase/protease
Alternative Names AF-1890; Diclondazolic Acid; DICA
CAS 50264-69-2
Storage -20°C, 3 years; 4°C, 2 years (Powder)
MWT 321.16
Solubility DMSO : 50 mg/mL (ultrasonic)
Clinical Information Phase 3
Target Apoptosis;Hexokinase;Mitochondrial Metabolism;Parasite
Applications
Application: Cancer-Kinase/protease

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